1-(AMINOALKYL)-3-SULFONYLAZAINDOLES AS LIGANDS FOR 5-HYDROXYTRYPTAMINE-6 Russian patent published in 2008 - IPC C07D471/04 C07D519/00 A61K31/437 A61P25/00 A61P25/22 A61P25/28

Abstract RU 2315048 C2

FIELD: organic chemistry, medicine, pharmacy.

SUBSTANCE: invention relates to compounds of the formula (I) , methods for their synthesis and their using for therapeutic treatment of the nervous system disorders associated with 5-HT-6 receptor. Invention provides synthesis of novel biologically active substances of the formula (I) and pharmaceutical compositions based on thereof used in treatment of the nervous system disorders and controlled by 5-HT-6 receptors.

EFFECT: valuable medicinal properties of compounds and pharmaceutical compositions.

6 tbl, 82 ex

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RU 2 315 048 C2

Authors

Bernotas Ronal'D Charl'Z

Lenisek Stiven Ehdvard

Antane Shujler A.

Dates

2008-01-20—Published

2003-06-03—Filed