IMPROVED PEPTIDE GASTRIN-RELEASING COMPOUNDS Russian patent published in 2008 - IPC C07K7/06 C07K14/595 A61K51/08 A61K49/00 

Abstract RU 2330859 C2

FIELD: chemistry.

SUBSTANCE: invention concerns compounds of the formula M-N-O-P-G, where M is a metal-chelating agent (in a complex with a radioactive metal nuclide or not), N-O-P is a linker, and G is a peptide for target transportation to a GRP receptor. Also the invention concerns methods of visualisation for a patient with the help of the claimed compounds, methods of obtaining a diagnostic visualisation and radiotherapeutic medium.

EFFECT: improved compounds for application in diagnostics visualisation or therapy.

49 cl, 51 dwg, 8 tbl, 58 ex

Similar patents RU2330859C2

Title Year Author Number
BLOOD DEPOT AGENTS FOR MAKING NUCLEAR MAGNETIC RESONANCE DIAGNOSIS 1999
  • Anelli P'Er Luchio
  • Brokketta Marino
  • De Khaen Kristof
  • Gatstsotti Ornella
  • Lattuada Luchano
  • Luks Dzhovanna
  • Manfredi Dzhuzeppe
  • Morozini P'Erfranchesko
  • Palano Daniela
  • Serleti Mikele
  • Uggeri Ful'Vio
  • Vizigalli Massimo
RU2250765C2
METHOD OF PRODUCING GAMMA AMIDES OF GLUTAMIC ACID 1999
  • Anelli P'Er Luchio
  • Brokketta Marino
  • De Khaen Kristof
  • Gatstsotti Ornella
  • Lattuada Luchano
  • Luks Dzhovanna
  • Manfredi Dzhuzeppe
  • Morozini P'Erfranchesko
  • Palano Daniela
  • Serleti Mikele
  • Uggeri Ful'Vio
  • Vizigalli Massimo
RU2395490C2
PEPTIDE VECTORS 2004
  • Dong Chzhen Ksin
  • Shen Jilana
  • Komstok Dzhinn Mehri
  • Kim San Kh.
RU2361876C2
FGF21 DERIVATIVES AND USE THEREOF 2015
  • Vechorek Birgit
  • Tagmose Tina Meller
  • Sass-Erum Kristian
  • Andersen Birgitta
  • Olsen Jergen
RU2729011C2
METHOD OF OBTAINING PEPTIDES 0
  • Nedamparambil A.Abrakham
  • Gans Veli Immer
  • Verner Robert Nelson
  • Kazimir Sestandzh
SU639446A3
ANALOGUES OF EGF(A) WITH SUBSTITUENTS-FATTY ACIDS 2017
  • Chen, Dzyankhe
  • Lau, Jesper F.
  • Kodra, Yanosh Tibor
  • Vechorek, Birgit
  • Linderot, Lars
  • Tegersen, Khenning
  • Rasmussen, Salka Elbel
  • Geribej, Patrik Uillyam
RU2747877C2
METHOD FOR PRODUCING BOC-THZ-PHE-D-TRP-LYS(BOC)-THR-NHCHCHNH-DOTA CONJUGATE BEING A PRECURSOR FOR ANTI-TUMOR RADIOPHARMACEUTICS 2022
  • Egorova Bajirta Vladimirovna
  • Fedotova Anzhelika Olegovna
  • Kolotaev Anton Vladimirovich
  • Osipov Vasilij Nikolaevich
  • Khachatryan Derenik Sarkisovich
RU2795447C1
METHOD OF PREPARING TETRADECAPEPTIDE 0
  • Dzhejms Edvin Shilds
SU904519A3
CONJUGATE INCLUDING LIGAND, SPACER, PEPTIDE LINKER AND BIOMOLECULE 2020
  • Akaiwa, Michinori
  • Ishida, Junya
  • Toya, Hiroki
  • Asano, Toru
  • Yoshikawa, Tomoaki
  • Sano, Yorikata
  • Sugano, Yukihito
RU2807081C2
METHOD OF SYNTHESIS OF MEMBRANE-BOUND COMPOUNDS 0
  • Gyunter Yung
  • Karl-Khajnts Vismyuller
  • Jerg Metsger
  • Khans-Ierg Byuring
  • Gerkhard Beker
  • Volfgang Besler
SU1823876A3

RU 2 330 859 C2

Authors

Kappelletti Ehnriko

Lattuada Luchiano

Linder Karen Eh.

Marinelli Ehdmund

Nan'Dzhappan Palaniappa

Radzhu Natarajan

Svenson Rol'F Eh.

Tvidl Majkl

Dates

2008-08-10Published

2003-12-24Filed