ARYLCARBONYL DERIVATIVES AS THERAPEUTIC AGENTS Russian patent published in 2008 - IPC C07D277/46 C07D417/04 C07D417/08 

Abstract RU 2340605 C2

FIELD: chemistry.

SUBSTANCE: in formula (Ib) R24 is selected from group, consisting of halogen, -CF3, -OCF3, -OR2, C1-6-alkyl-Z- and R6-W1-C1-6alkylene-Z-; L1 is bond, -O-, -S-, -S(O)2-, -C(O)- or -N(R11)-; G1 is C1-6-alkyl, C3-10-cycloalkyl or piperidyl, optionally substituted with one or several substituents, selected from C3-10-cycloalkyl, L2 is -N(R20)-; L3 is -C(O)-; R1 is hydrogen; G2 is .

EFFECT: increase of composition and treatment method efficiency.

33 cl, 15 dwg, 480 ex

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RU 2 340 605 C2

Authors

Polizetti Dkharma Rao

Kodra Janos Tibor

Lau Jesper

Blok Pav

Val'Karse-Lopes Marija Karmen

Blume Nil'S

Guzel' Mustafa

Santosh Kalpati Chidambaresvaran

Mdzhalli Adnan M. M.

Ehndrjus Robert Karl

Subramanian Govindan

Ankersen Mikhael'

Vedse Per

Mjurrehj Ehntoni

Jeppesen Lone

Lau Jesper

Dates

2008-12-10Published

2003-06-27Filed