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2 368 613

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(51)

IPC

C07D451/04(2006-01-01)

A61K31/46(2006-01-01)

A61P29/00(2006-01-01)

(21) (22)

Application

2008105923/04, 2008-02-19

(24)

Start date

2008-02-19

(22)

Actual filing date

2008-02-19

(45)

Published

2009-09-27

(72)

Inventor

Shevchenko Valerij PavlovichMjasoedov Nikolaj FedorovichNagaev Igor' Julianovich

(73)

Holder

Institut Molekuljarnoj Genetiki Rossijskoj Akademii Nauk Ran) Gosudarstvennogo Uchrezhdenija)

UNIFORMLY TRITIUM-LABELED 4,4-DIFLUORO-N-{(1S)-3-[3-(3-ISOPROPYL-5-METHYL-4H-1,2,4-TRIAZOL-4-YL)-8-AZABICYCLO[3,2,1]OCT-8-YL]-1-PHENYLPROPYL}CYCLOHEXANE CARBODIIMIDE Russian patent published in 2009 - IPC C07D451/04 A61K31/46 A61P29/00

Abstract RU 2368613 C1

FIELD: chemistry.

SUBSTANCE: described is a new uniformly tritium-labeled 4,4-fluoro-N-{(1S)-3-[3-(3-isopropyl-5-methyl-4H-1,2,4-trizol-4-yl)-8-azabicyclo[3.2.1]oct-8-yl]-1-phenylpropyl}cyclohexane carboiimide (maraviroc) of formula I .

EFFECT: said compound can be used in analysis of physiologically active compound-analogue.

1 cl, 1 ex, 2 dwg

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RU 2 368 613 C1

Authors

Shevchenko Valerij Pavlovich

Mjasoedov Nikolaj Fedorovich

Nagaev Igor' Julianovich

Dates

2009-09-27—Published

2008-02-19—Filed