PHARMACEUTICAL COMPOSITIONS CONTAINING MIRTAZAPIN SALT Russian patent published in 2009 - IPC C07D471/14 A61K31/55 A61P25/24 

Abstract RU 2375362 C2

FIELD: medicine.

SUBSTANCE: invention refers to method for prevention of mirtazapin sublimation from a pharmaceutical preparative form containing solid enantiomer pure form of mirtazapin, by making the preparative forms by addition of at least one pharmaceutically acceptable adjuvant to the solid form of mirtazapin enantiomer. The enantiomer pure form is pharmaceutically acceptable, nonsublumating and solid salt of S- or R-mirtazapin. There are also described nonsublumating salts of S-mirtazapin and the pharmaceutical preparative form of the latter.

EFFECT: higher efficiency of the composition.

4 cl, 4 tbl, 8 ex

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RU 2 375 362 C2

Authors

Molenar Sitske Khike

Kemperman Gerardus Jokhannes

Van Der Vort Marsalk Kes

Dates

2009-12-10Published

2005-04-19Filed