STEREOSELECTIVE SYNTHESIS OF VITAMINE D ANALOGUES Russian patent published in 2010 - IPC C07C401/00 

Abstract RU 2380359 C2

FIELD: chemistry.

SUBSTANCE: present invention relates to intermediate compounds used in synthesis of calcipotriol or monohydrate of calcipotriol, to methods of synthesising said intermediate compounds and to methods for stereoselective reduction of the said intermediate compounds.

EFFECT: method increases output of C-24 hydroxy epimers of calciprotriol derivatives.

27 cl, 16 ex, 1 tbl

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RU 2 380 359 C2

Authors

Sabro Tomas Peter

Kelverli Martin Dzhon

Dates

2010-01-27Published

2005-03-10Filed