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2 382 789

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IPC

C07D498/04(2006-01-01)

A61K31/538(2006-01-01)

(21) (22)

Application

2006142705/04, 2005-05-04

(24)

Start date

2005-05-04

(22)

Actual filing date

2005-05-04

(45)

Published

2010-02-27

(72)

Inventor

Takhri AbdellakhMikhils Liv Ehmma JanVan Akker Kunrad Lodevejk AugustSjurlero Dominik Lui Nestor Gilehjn

(73)

Holder

Tibotek Farmas'Jutikalz Ltd.

DERIVATIVES OF 1,10b-DIHYDRO-2-(AMINOCARBONYLPHENYL)-5H-PYRAZOLO[1,5-c][1,3]BENZOXASIN-5-YL)PHENYLMETHYLMETHANON AS INHIBITORS OF HIV VIRUS REPLICATION Russian patent published in 2010 - IPC C07D498/04 A61K31/538

Abstract RU 2382789 C2

FIELD: medicine, pharmaceutics.

SUBSTANCE: described are derivatives of 5H-pyrazolo[1,5-c][1,3]benzoxasin-5-yl)phenylmethanon of formula , possessing ability to inhibit HIV replication, where values of R¹, R², R³ substitutes are given in invention formula. Also describes is pharmaceutical preparation and application of compound for obtaining medication applied for treatment of conditions associated with HIV infection.

EFFECT: claimed compounds are applicable for prevention or treatment of HIV-produced infection and for AIDS treatment.

15 cl, 3 tbl, 5 ex

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RU 2 382 789 C2

Authors

Takhri Abdellakh

Mikhils Liv Ehmma Jan

Van Akker Kunrad Lodevejk August

Sjurlero Dominik Lui Nestor Gilehjn

Dates

2010-02-27—Published

2005-05-04—Filed