DERIVATIVES OF 1,10b-DIHYDRO-2-(AMINOCARBONYLPHENYL)-5H-PYRAZOLO[1,5-c][1,3]BENZOXASIN-5-YL)PHENYLMETHYLMETHANON AS INHIBITORS OF HIV VIRUS REPLICATION Russian patent published in 2010 - IPC C07D498/04 A61K31/538 

Abstract RU 2382789 C2

FIELD: medicine, pharmaceutics.

SUBSTANCE: described are derivatives of 5H-pyrazolo[1,5-c][1,3]benzoxasin-5-yl)phenylmethanon of formula , possessing ability to inhibit HIV replication, where values of R1, R2, R3 substitutes are given in invention formula. Also describes is pharmaceutical preparation and application of compound for obtaining medication applied for treatment of conditions associated with HIV infection.

EFFECT: claimed compounds are applicable for prevention or treatment of HIV-produced infection and for AIDS treatment.

15 cl, 3 tbl, 5 ex

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RU 2 382 789 C2

Authors

Takhri Abdellakh

Mikhils Liv Ehmma Jan

Van Akker Kunrad Lodevejk August

Sjurlero Dominik Lui Nestor Gilehjn

Dates

2010-02-27Published

2005-05-04Filed