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(19)

(11)

2 416 615

(13)

(51)

IPC

C07D498/04(2006-01-01)

A61K31/5365(2006-01-01)

A61P31/18(2006-01-01)

(21) (22)

Application

2007141639/04, 2006-04-11

(24)

Start date

2006-04-11

(22)

Actual filing date

2006-04-11

(45)

Published

2011-04-20

(72)

Inventor

Takhri AbdellakhKhu LiliSjurlero Dominik Lui Nestor GilehjnVigerink Pit Tom Bert Pol'

(73)

Holder

Tibotek Farmas'Jutikalz Ltd.

(1,10b-DIHYDRO-2-(AMINOALKYLPHENYL)-5H-PYRAZOLO[1,5-c][1,3] BENZOXAZIN-5-YL) PHENYLMETHANONE DERIVATIVES AS HIV VIRAL REPLICATION INHIBITORS Russian patent published in 2011 - IPC C07D498/04 A61K31/5365 A61P31/18

Abstract RU 2416615 C2

FIELD: chemistry.

SUBSTANCE: invention relates to (5H-pyrazolo[1,5-c][1,3]benzoxazin-5-yl)phenylmethanone derivatives (I), useful as HIV viral replication inhibitors, as well as pharmaceutical compositions, use thereof as medicinal agents.

EFFECT: disclosed compounds are meant for preventing or treating HIV infection and treating AIDS.

7 cl, 2 tbl, 4 ex

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RU 2 416 615 C2

Authors

Takhri Abdellakh

Khu Lili

Sjurlero Dominik Lui Nestor Gilehjn

Vigerink Pit Tom Bert Pol'

Dates

2011-04-20—Published

2006-04-11—Filed