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2 396 263

(13)

(51)

IPC

C07D285/135(2006-01-01)

A61K31/433(2006-01-01)

A61P29/00(2006-01-01)

(21) (22)

Application

2008129503/04, 2008-07-17

(24)

Start date

2008-07-17

(22)

Actual filing date

2008-07-17

(45)

Published

2010-08-10

(72)

Inventor

Pulina Natal'Ja AlekseevnaJushkov Vladimir ViktorovichSobin Fedor VladimirovichJatsenko Konstantin VjacheslavovichZalesov Vladimir Vasil'Evich

(73)

Holder

Gosudarstvennoe Obrazovatel'Noe Uchrezhdenie Vysshego Professional'Nogo Obrazovanija Gosudarstvennaja Farmatsevticheskaja Akademija Federal'Nogo Agentstva Po Zdravookhraneniju I Sotsial'Nomu Razvitiju" Vpo Pgfa Roszdrava)

BIS{3-PHENYL-1-[2-(5-METHYL-1,3,4-THIADIAZOLYL)]CARBOXAMIDO-1,3-PROPANEDIONATO}MANGANESE HAVING ANTI-INFLAMMATORY AND ANALGESIC ACTVITY Russian patent published in 2010 - IPC C07D285/135 A61K31/433 A61P29/00

Abstract RU 2396263 C2

FIELD: chemistry.

SUBSTANCE: invention relates to organic chemistry and specifically to novel biologically active substances of the class of complex compounds of N-heterylamides of 4-aryl-2,4-dioxobutanoic acids. The invention discloses bis{3-phenyl-1-[2-(5-methyl-1,3,4-thiadiazolyl)]carboxamido-1,3-propanedionato}manganese having anti-inflammatory and analgesic activity and formula: .

EFFECT: high output of compounds with pronounced anti-inflammatory and analgesic activity, as well as low toxicity.

1 cl, 1 tbl, 1 ex

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RU 2 396 263 C2

Authors

Pulina Natal'Ja Alekseevna

Jushkov Vladimir Viktorovich

Sobin Fedor Vladimirovich

Jatsenko Konstantin Vjacheslavovich

Zalesov Vladimir Vasil'Evich

Dates

2010-08-10—Published

2008-07-17—Filed