FIELD: medicine, pharmaceutics.
SUBSTANCE: there are described compounds of formula I: , their pharmaceutically acceptable salts where R1-R7, Y and n are specified in the patent claim. The compounds exhibit inhibitory action in the relation to aurora A tyrosine kinase. There is also described a drug of the compound of formula (I). The drug can be used for control or prevention of diseases, such as cancer.
EFFECT: preparation of new phthalazinone derivatives which can be used for control or prevention of diseases, such as cancer.
17 cl, 2 tbl, 41 ex
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Authors
Dates
2010-08-20—Published
2005-09-23—Filed