KAPPA-OPIOID AGONIST Russian patent published in 2011 - IPC A61K31/4188 

Abstract RU 2413512 C1

FIELD: medicine, pharmaceutics.

SUBSTANCE: invention refers to drugs and concerns application of 9-dialkylaminoethylsubsituted-2-(4-fluorophenyl)imidazo[1,2]benzimidazole dihydrochloride of general formula I (where NR2 has the values specified in the formula) as a kappa-opioid the agonist.

EFFECT: invention aims at extending the range of products exhibiting kappa-opioid agonistic activity.

2 tbl, 3 ex

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Authors

Spasov Aleksandr Alekseevich

Anisimova Vera Alekseevna

Vasil'Ev Pavel Mikhajlovich

Grechko Olesja Jur'Evna

Eliseeva Natal'Ja Vladimirovna

Tolpygin Ivan Evgen'Evich

Minkin Vladimir Isaakovich

Dates

2011-03-10Published

2009-07-29Filed