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2 572 711

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IPC

A61K31/4188(2006-01-01)

A61P21/02(2006-01-01)

A61K31/5375(2006-01-01)

(21) (22)

Application

2014137853/15, 2014-09-19

(24)

Start date

2014-09-19

(22)

Actual filing date

2014-09-19

(45)

Published

2016-01-20

(72)

Inventor

Spasov Aleksandr AlekseevichPetrov Vladimir IvanovichAnisimova Vera AlekseevnaMinkin Vladimir IsaakovichSukhov Aleksandr GeorgievichGrechko Olesja Jur'EvnaMatukhno Aleksej Evgen'EvichKalitin Konstantin Jur'Evich

(73)

Holder

Federal'Noe Gosudarstvennoe Avtonomnoe Obrazovatel'Noe Uchrezhdenie Vysshego Obrazovanija Federal'Nyj Universitet"Gosudarstvennoe Bjudzhetnoe Obrazovatel'Noe Uchrezhdenie Vysshego Professional'Nogo Obrazovanija Gosudarstvennyj Meditsinskij Universitet" Ministerstva Zdravookhranenija Rossijskoj Federatsii

ANTICONVULSANT Russian patent published in 2016 - IPC A61K31/4188 A61P21/02 A61K31/5375

Abstract RU 2572711 C1

FIELD: medicine.

SUBSTANCE: method is implemented by using 9-dialkyl aminoethyl-2-(4-fluorophenyl)imidazo[1,2-a]-benzimidazole dihydrochloride of general formula I , wherein a) NR₂ = pyrrolidino; b) NR₂ = morpholino as an agent possessing anticonvulsant activity. The compound may be used for preparing an anticonvulsant.

EFFECT: higher anticonvulsant activity.

2 cl, 8 dwg, 1 tbl

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RU 2 572 711 C1

Authors

Spasov Aleksandr Alekseevich

Petrov Vladimir Ivanovich

Anisimova Vera Alekseevna

Minkin Vladimir Isaakovich

Sukhov Aleksandr Georgievich

Grechko Olesja Jur'Evna

Matukhno Aleksej Evgen'Evich

Kalitin Konstantin Jur'Evich

Dates

2016-01-20—Published

2014-09-19—Filed