FIELD: medicine, pharmaceutics.
SUBSTANCE: given invention refers to pharmacology and concerns a pharmaceutical composition for increasing nitrogen oxide release from human endotheliocytes, containing at least one diastereoisomer of glucuronidated nebivolol metabolite of formula
as well as to a standard dosage form containing at least at least one diastereoisomer of glucuronidated nebivolol metabolite of formula 1.
EFFECT: invention provides effective nitrogen oxide release and facilitated washout of nebivolol metabolites.
2 cl, 5 dwg, 4 tbl, 1 ex
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Authors
Dates
2011-03-10—Published
2006-01-30—Filed