FIELD: chemistry.
SUBSTANCE: invention relates to indol-3-yl-carbonyl-spiro-piperadine derivatives used as V1a receptor antagonists and which have formula I: , where the spiro-piperadine A head group and residues R1, R2 and R3 are as defined in claim 1 of the invention. The invention also pertains to pharmaceutical compositions which contain such compounds and use thereof in preparing medicines with V1a receptor antagonist activity.
EFFECT: high activity of derivatives.
37 cl, 1 tbl, 285 ex
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Authors
Dates
2011-03-20—Published
2006-07-04—Filed