INDOLE-3-YL-CARBONYL-PIPERIDINE AND PIPERAZINE DERIVATIVES Russian patent published in 2011 - IPC C07D401/06 C07D401/14 C07D403/06 C07D405/02 A61K31/404 A61K31/454 

Abstract RU 2422442 C2

FIELD: medicine, pharmaceutics.

SUBSTANCE: invention refers to new indole-3-yl-carbonyl-piperidine and piperazine derivatives of formula I: where the values R1 R2 R3, A are presented in the claim 1.

EFFECT: compounds exhibit antagonist activity thereby applicable in a pharmaceutical composition.

20 cl, 230 ex

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Authors

Bissants Katerina

Grundshober Kristof

Ratni Khasan

Rodzhers-Ehvans Mark

Shnajder Patrik

Dates

2011-06-27Published

2006-07-19Filed