FIELD: medicine.
SUBSTANCE: invention refers to indole-3-yl-carbonyl-spiro-piperidine derivatives which have an effect of Vla-receptor antagonists and are presented by Formula I:
where a tail spiropiperidine group A and residual R1, R2 and R3 are such as specified in the patent claim.
EFFECT: higher efficiency of applying the compounds in drugs effective in dysmenorrhea, hypertension, chronic heart failure, inadequate vasopressin secretion, hepatic cirrhosis, nephrotic syndrome, obsessive-compulsive disorder, anxious and depressive disorders.
22 cl, 42 ex
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Authors
Dates
2011-06-10—Published
2006-12-19—Filed