FIELD: medicine, pharmaceutics.
SUBSTANCE: invention refers to new cyclopenta[b]benzofuranyl derivatives of formula 
wherein substitutes R1, R2, R3, R4, R5, R6 and R7 and n are specified in the patent clam. These compounds exhibit properties of NF-kB-activity and/or AP-1 inhibitor/modulator. Also, the inventive subject matter are methods for preparing intermediate compounds thereof, a pharmaceutical composition containing them, administration thereof for prevention and/or treatment of inflammatory and autoimmune diseases, neurodegenerative diseases and hyperproliferative diseases caused by NF-kB- and/or AP-1-activity, and a method for prevention and/or treatment of said diseases.
EFFECT: preparation of new cyclopenta[b]benzofuranyl derivatives.
21 cl, 3 tbl, 151 ex
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