APPLICATION OF THIENOPYRIDONE DERIVATIVES AS AMPA-ACTIVATORS AND PHARMACEUTIC COMPOSITIONS, CONTAINING THEM Russian patent published in 2011 - IPC A61K31/4436 C07D495/04 A61P3/10 

FIELD: medicine, pharmaceutics.

SUBSTANCE: invention relates to application of thienopyridone derivatives of formula (I), in which B represents CH, represents , or , R represents H, R¹ and R², independently on each other, represent H, linear or branched (C₁-C₄)alkyl, (C1-C₄)cycloalkyl, halogen or together form group -(CH₂)_n-, where n=1- 4, R³ and R⁴, independently on each other, represent H, R⁶ represents H, X represents -O-, or their pharmaceutically acceptable salts for preparation of pharmaceutical composition.

EFFECT: obtaining pharmaceutical composition, suitable for treatment of diabetes, metabolic syndrome and obesity.

8 cl, 1 tbl, 210 ex