OXAZINMONOACYLGLYCERIN LIPASE (MAGL) INHIBITORS Russian patent published in 2023 - IPC C07D498/04 A61K31/5375 A61P25/00 A61P29/00 A61P35/00 

Abstract RU 2794334 C2

FIELD: medicine.

SUBSTANCE: invention relates to new heterocyclic compounds having the general formula (Ic), as well as to compositions comprising these compounds, methods for the manufacture of these compounds and methods of using these compounds.

EFFECT: new compounds have been obtained that can be used to inhibit the activity of monoacylglycerol lipase (MAGL).

44 cl, 3 tbl, 2 ex

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RU 2 794 334 C2

Authors

Bell, Charlz

Bents, Jerg

Gobbi, Luka

Greter, Uve

Grebke Tsbinden, Katrin

Khansen, Dennis Zhyul

Khornsperger, Benua

Kotser, Byulent

Kroll, Karsten

Kun, Bernd

O'Khara, Fionn

Rikhter, Khans

Ritter, Martin

Tsutiya, Satosi

Chen, Zhuj

Dates

2023-04-17Published

2019-03-22Filed