FIELD: chemistry.
SUBSTANCE: invention relates to novel oxadiazole compounds of formula
(1) and pharmaceutically acceptable salts thereof, where R1 and R2 assume values given in the description, Y is a single bond. The invention also relates to use of said compounds as DGAT1 inhibitors, for example for treating obesity and diabetes, and a method of inhibiting.
EFFECT: high treatment efficiency.
13 cl, 65 tbl, 712 ex
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Authors
Dates
2011-06-20—Published
2005-12-09—Filed