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2 624 021

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(51)

IPC

C07D495/04(2006-01-01)

A61K31/519(2006-01-01)

A61P3/10(2006-01-01)

(21) (22)

Application

2014126341, 2012-10-23

(24)

Start date

2012-10-23

(22)

Actual filing date

2012-10-23

(45)

Published

2017-06-30

(72)

Inventor

Lyu KhunLi TszyaLi TszyanLi TszingyaVan TszyanSu MinboLyan TszeTszyan KhualyanChen Kajsyan

(73)

Holder

Shankhaj Instityut Of Matiria Medika, Chajniz Ekedemi Of SajensizTsyzen Farmasyutikal Ko., Ltd.

COMPOUNDS OF THIENYL[3, 2-d]PYRIMIDINE-4-ON, METHOD FOR PRODUCTION, PHARMACEUTICAL COMPOSITIONS AND THEIR APPLICATION Russian patent published in 2017 - IPC C07D495/04 A61K31/519 A61P3/10

Abstract RU 2624021 C2

FIELD: pharmacology.

SUBSTANCE: invention relates to new compounds of thienyl[3,2-d] pyrimidin-4-on of general formula pharmaceutical compositions based thereon and their pharmacological applications.

EFFECT: new compounds that are inhibitors of DPPIV, which can be used as medicaments for diabetes treatment, have been obtained.

15 cl, 12 tbl, 149 ex, 13 dwg

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RU 2 624 021 C2

Authors

Lyu Khun

Li Tszya

Li Tszyan

Li Tszingya

Van Tszyan

Su Minbo

Lyan Tsze

Tszyan Khualyan

Chen Kajsyan

Dates

2017-06-30—Published

2012-10-23—Filed