AMIDOACETONITRILE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING SAID DERIVATIVES AND USE THEREOF IN PREPARING MEDICINAL AGENT Russian patent published in 2011 - IPC C07C381/00 A01N41/12 A01P5/00 

Abstract RU 2425825 C2

FIELD: chemistry.

SUBSTANCE: invention relates to compounds of formula

or a tautomer or prodrug, or a pharmaceutically acceptable salt of the said compound, tautomer or prodrug, where each of R1, R2, R3, R4 and R5 is independently selected from H, halogen, CN, CF3 and CONH2; and compositions containing said compounds, and use of said compositions as antiparasite agents.

EFFECT: high effectiveness of the compounds.

11 cl, 74 ex

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RU 2 425 825 C2

Authors

Komlehj Stjuart Nikolas

Khannam Dzhoanna Klehr

Khouson Uill'Jam

Lore Kristell'

Sabnis Jodzhesh Anil

Dates

2011-08-10Published

2008-01-29Filed