DERIVATIVES OF SUBSTITUTED 3-SULPHONYLINDAZOLE AS 5-HYDROXYTRYPTAMINE-6 LIGANDS Russian patent published in 2011 - IPC C07D231/56 C07D403/12 A61K31/416 A61P25/28 

Abstract RU 2429231 C2

FIELD: chemistry.

SUBSTANCE: invention discloses a compound of formula I

, in which radicals and groups are described in the claims. Said compounds are 5-hydroxytryptamine-6 (5-HT6) ligands and can be used to treat central nervous system disorders associated with or influenced by the 5-HT6 receptor. The invention also relates to a pharmaceutical composition and a method of treating said disorders.

EFFECT: high efficiency of using said derivatives.

19 cl, 13 tbl, 204 ex

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RU 2 429 231 C2

Authors

Ehlokdakh Khasan Makhmud

Grinfild Aleksandr Aleksej

L'Ju Kevin

Makdevit Robert Ehmmet

Makfarlehjn Dzheral'Din Rut

Grosanu Kristina

Lo Dzhenifer Rebekka

Li Janfang

Robichaud Al'Bert Dzhen

Bernotas Ronal'D Charl'Z

Dates

2011-09-20Published

2006-08-08Filed