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(19)

RU

(11)

2 621 052

(13)

C2

(51)

IPC

C07D295/14(2006-01-01)

C07D405/12(2006-01-01)

C07D405/14(2006-01-01)

A61K31/453(2006-01-01)

A61K31/46(2006-01-01)

A61K31/496(2006-01-01)

A61K31/5377(2006-01-01)

A61P35/00(2006-01-01)

(21) (22)

Application

2013133800, 2013-07-19

(24)

Start date

2009-12-04

(22)

Actual filing date

2013-07-19

(45)

Published

2017-05-31

(72)

Inventor

Branko MilanDin KhunDouerti Dzhordzh A.Elmor Stiven V.Khasvold LizaKheksamer LauraKanzer Aaron R.Mantej Robert A.Makklellan Uillyam Dzh.Park Chang Kh.Park Cheol-MinPetros Endryu M.Sun SyaokhunSauers Endryu Dzh.Sallivan Dzherard M.Tao Chzhi-FuVan Gari T.Van LeVan SiluUendt Majkl D.

(73)

Holder

Ebbvi Ink.

APOPTOSIS INDUCING AGENTS SELECTIVE FOR Bcl-2 FOR CANCER AND IMMUNE DISEASES TREATMENT Russian patent published in 2017 - IPC C07D295/14 C07D405/12 C07D405/14 A61K31/453 A61K31/46 A61K31/496 A61K31/5377 A61P35/00 

Abstract RU 2621052 C2

FIELD: pharmacy.

SUBSTANCE: invention relates to specific heterocyclic compounds containing the sulphonyl amino carbonyl group. The invention also relates to a pharmaceutical composition based on this compound.

EFFECT: new heterocyclic compounds with inhibitory activity in terms of anti-apoptotic Bcl-2 proteins are obtained.

2 cl, 3 tbl, 481 ex

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RU 2 621 052 C2

Authors

Branko Milan

Din Khun

Douerti Dzhordzh A.

Elmor Stiven V.

Khasvold Liza

Kheksamer Laura

Kanzer Aaron R.

Mantej Robert A.

Makklellan Uillyam Dzh.

Park Chang Kh.

Park Cheol-Min

Petros Endryu M.

Sun Syaokhun

Sauers Endryu Dzh.

Sallivan Dzherard M.

Tao Chzhi-Fu

Van Gari T.

Van Le

Van Silu

Uendt Majkl D.

Dates

2017-05-31—Published

2013-07-19—Filed

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