5-AMINO-3-(2-NITROXIPROPYL)-1,2,4-THIADIAZOLES Russian patent published in 2011 - IPC C07D285/08 C07D285/135 C07D417/04 A61K31/433 A61K31/4523 A61P25/28 

Abstract RU 2434856 C1

FIELD: medicine, pharmaceutics.

SUBSTANCE: invention relates to derivatives of 5-amino-3-(2-nitroxipropyl)-1,2,4-thiadiazoles of general formula , where R1, R2 can be similar or different and independently represent hydrogen, substituted or non-substituted aryl or heteroaryl or aralkyl, alkyl, cycloalkyl, and R1 + R2 can represent heteroaryl (optionally substituted piperasin and piperidin).

EFFECT: obtained are novel compounds, which can be applied in medicine for treatment of neurodegenerative diseases.

1 cl, 3 ex

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RU 2 434 856 C1

Authors

Proshin Aleksej Nikolaevich

Serkov Igor' Viktorovich

Bachurin Sergej Olegovich

Dates

2011-11-27Published

2010-10-15Filed