OLIGOPEPTIDE HAVING NEUREGULIN-1 ACTIVITY ON CARDIOMYOCYTE PROLIFERATION Russian patent published in 2012 - IPC C07K7/06 A61K38/08 A61P9/00 

Abstract RU 2439078 C1

FIELD: chemistry.

SUBSTANCE: method is realised by forming an oligopeptide having neuregulin-1 activity on cardiomyocyte proliferation, said oligopeptide having general formula: X1-X2-X3-X4-X5-X6-X7, where X1 is K, X2 is G or A, X3 is A or is absent, X4 is M, X5 is G or A, X6 is A or is absent, X7 is K, where the size of the oligopeptide varies from penta to heptapeptide.

EFFECT: obtaining a synthetic analogue of neuregulin-1 growth factor, capable of stimulating cardiomyocyte proliferation as a result of binding with receptors on the surface of stem cells.

2 dwg, 2 ex

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RU 2 439 078 C1

Authors

Golubovich Vladimir Petrovich

Gribovskaja Ol'Ga Viktorovna

Shutova Irina Vladimirovna

Goranov Vitalij Anatol'Evich

Kovalenko Aleksandr Pavlovich

Dates

2012-01-10Published

2010-08-02Filed