Show metadata Hide metadata

(19)

(11)

2 440 351

(13)

(51)

IPC

C07D487/04(2006-01-01)

A61K31/4192(2006-01-01)

A61K31/53(2006-01-01)

A61P37/02(2006-01-01)

(21) (22)

Application

2008127502/04, 2006-12-05

(24)

Start date

2006-12-05

(22)

Actual filing date

2006-12-05

(45)

Published

2012-01-20

(72)

Inventor

Geda FilippBuassi GijomBor-Kapra KatrinKollan FrederikDav'E LoranFormstesher Eht'EnnZhak Ksav'ERehn Zhan-KristofDelansorn RemiPeretto IlariaVin'Jando Stefano

(73)

Holder

Ibrizheniks Sa

NOVEL CYSTEINE PROTEASE INHIBITORS, PHARMACEUTICAL COMPOSITIONS THEREOF AND THERAPEUTIC APPLICATION THEREOF Russian patent published in 2012 - IPC C07D487/04 A61K31/4192 A61K31/53 A61P37/02

Abstract RU 2440351 C2

FIELD: chemistry.

SUBSTANCE: invention describes novel compounds of general formula in which is or (values of radicals are given in the claim), a method of producing said compounds, a pharmaceutical composition containing said compounds and therapeutic application thereof.

EFFECT: compounds are cysteine protease inhibitors and can be used in medicine.

25 cl, 1 tbl, 41 ex

Similar patents RU2440351C2

Title	Year	Author	Number
NEW TETRACYCLIC CYSTEIN PROTEASE INHIBITORS, PHARMACEUTICAL COMPOSITIONS THEREOF AND APPLICATION THEREOF	2007	Geda Filipp Zhak Ksav'E Kollan Frederik Dav'E Loran Formstesher Eht'Enn Rehn Zhan-Kristof Kolombo Matteo	RU2481349C2
NOVEL CYSTEINE PROTEASE INHIBITORS AND THERAPEUTIC APPLICATION THEREOF	2006	Geda Filipp Buassi Gijom Bor-Kapra Katrin Kollan Frederik Dav'E Loran Formstesher Eht'Enn Zhak Ksav'E Rehn Zhan-Kristof Delansorn Remi Valleze Stefanija Kolombo Matteo	RU2424234C2
SELECTIVE AND REVERSIBLE UBIQUITIN-SPECIFIC PROTEASE 7 INHIBITOR	2012	Kollan Frederik Gurdel Mari-Edit	RU2622640C2
BENZOFURAN DERIVATIVES	2004	Sato Sejiti Kosi Tomojuki Mizoguti Tosimi Jasuoka Kioko Kumai Natsujo Totsuka Dzunko Tamura Masakhiro Okhkuti Masao	RU2328495C2
PEPTIDE MACROCYCLES AGAINST ACINETOBACTER BAUMANNII	2019	Blajger, Konrad Cheang, Daniella Di Dzhordzho, Patrik Khu, Tajshan Jenni, Kristian Mattej, Patritsio Shmits, Petra Shtoll, Teodor	RU2795374C2
METHOD OF SYNTHESIS OF DERIVATIVE OF 8-CYCLO-PENTYL-6-ETHYL-3- (SUBSTITUTED)-5,8-DIHYDRO-4H-1,2,3A,7,8-PENTAAZA-AC-INDACENE (VARIANTS) AND INTERMEDIATE COMPOUNDS	2000	Urban Frehnk Dzhon	RU2189985C2
PEPTIDE MACROCYCLES AGAINST ACINETOBACTER BAUMANNII	2016	Alanin Aleksander Bene Zhyulen Blajger Konrad Fashing Bernard Khilpert Khans Khu Tajshan Makdonald Duajt Dzhekson Stiven Kolchevski Sabine Kroll Karsten Shojblin Adrian Shen Khun Shtoll Teodor Tomas Khelmut Vakhkhab Amal Tsampaloni Klaudia	RU2729609C2
DERIVATIVES OF BETA-AMINO ACID NITRILES	2001	Tobias Gabriel' Mikhaehl' Pekh Roza-Marija Rodriges-Sarm'Ento	RU2245871C2
DERIVATIVES OF PYRROLO[3,2-c]PYRIDIN-4-ONE 2-INDOLINONE AS PROTEINKINASE INHIBITORS	2007	Tan Pehn Cho Su Idun Chzhan Lehj Sjao Lu	RU2410387C2
DEVICES FOR BLOOD INTAKE, CONTAINING LYSOPHOSPHOLIPASE INHIBITOR	2012	Kraft Devid Ept Priyanka	RU2623049C2

RU 2 440 351 C2

Authors

Geda Filipp

Buassi Gijom

Bor-Kapra Katrin

Kollan Frederik

Dav'E Loran

Formstesher Eht'Enn

Zhak Ksav'E

Rehn Zhan-Kristof

Delansorn Remi

Peretto Ilaria

Vin'Jando Stefano

Dates

2012-01-20—Published

2006-12-05—Filed