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(19)

(11)

2 729 609

(13)

(51)

IPC

C07D513/04(2006-01-01)

C07D417/06(2006-01-01)

C07K5/02(2006-01-01)

A61K38/00(2006-01-01)

A61K31/04(2006-01-01)

(21) (22)

Application

2018113426, 2016-10-24

(24)

Start date

2016-10-24

(22)

Actual filing date

2016-10-24

(45)

Published

2020-08-11

(72)

Inventor

Alanin AleksanderBene ZhyulenBlajger KonradFashing BernardKhilpert KhansKhu TajshanMakdonald DuajtDzhekson StivenKolchevski SabineKroll KarstenShojblin AdrianShen KhunShtoll TeodorTomas KhelmutVakhkhab AmalTsampaloni Klaudia

(73)

Holder

F. Hoffmann-La Roche Ag

PEPTIDE MACROCYCLES AGAINST ACINETOBACTER BAUMANNII Russian patent published in 2020 - IPC C07D513/04 C07D417/06 C07K5/02 A61K38/00 A61K31/04

Abstract RU 2729609 C2

FIELD: medicine; pharmaceuticals.

SUBSTANCE: invention relates to novel compounds of formula (I), as well as to pharmaceutical compositions based thereon and use.

(I).

EFFECT: obtaining novel compounds which can be used as medicinal agents for treating diseases and infections caused by Acinetobacter baumannii.

22 cl, 5 tbl, 255 ex

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RU 2 729 609 C2

Authors

Alanin Aleksander

Bene Zhyulen

Blajger Konrad

Fashing Bernard

Khilpert Khans

Khu Tajshan

Makdonald Duajt

Dzhekson Stiven

Kolchevski Sabine

Kroll Karsten

Shojblin Adrian

Shen Khun

Shtoll Teodor

Tomas Khelmut

Vakhkhab Amal

Tsampaloni Klaudia

Dates

2020-08-11—Published

2016-10-24—Filed