FACTOR Xa INHIBITOR SALT, METHOD FOR MAKING IT, BASED PHARMACEUTICAL COMPOSITION, TABLET, CAPSULE AND LOZENGE CONSISTING OF THIS COMPOSITION, METHOD FOR TREATING THROMBOSIS AND METHOD FOR INHIBITING BLOOD SAMPLE COAGULATION Russian patent published in 2012 - IPC C07D213/75 A61K31/44 A61P7/02 

Abstract RU 2440986 C2

FIELD: medicine, pharmaceutics.

SUBSTANCE: invention refers to a factor Xa inhibitor salt containing a compound of structural formula I: and maleic acid. The invention also concerns a pharmaceutical composition, to a tablet, to a capsule, to a lozenge, to a method for preventing or treating a condition characterised by adverse thrombotic events in a mammal, to a method for inhibiting blood sample coagulation, as well as to a method for making the compound of structural formula I.

EFFECT: making the new biologically active compound for preventing or treating the condition characterised by adverse thrombotic events.

28 cl, 4 ex, 7 tbl, 6 dwg

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RU 2 440 986 C2

Authors

Grant Krejg

Kehnter Dzhejms P.

Lehnglehndz Grejehm

Dates

2012-01-27Published

2006-11-07Filed