PHARMACEUTICAL COMPOSITION POSSESSING ANTIINFLAMMATORY, BRONCHOLYTIC, ANTI-TUBERCULOSIS ACTIVITY Russian patent published in 2012 - IPC C07D285/135 A61K31/433 A61P29/00 

Abstract RU 2448961 C1

FIELD: medicine, pharmaceutics.

SUBSTANCE: invention relates to pharmaceutical composition possessing anti-inflammatory, broncholytic and anti-tuberculosis activity, which represents N-(5-ethyl-1,3,4-thiadiazole-2-yl)-4-nitrobenzamide. Obtained results of pharmacological study showed that claimed compound possesses high anti-inflammatory, broncholytic and anti-tuberculosis activity, which are not worse and in some cases is better than known applied in medicine preparations. Elaborated is solid dosed pharmaceutical composition based on claimed compound, made in form of tablets, or capsules, or in form of powder for preparation of suspension for drinking.

EFFECT: obtaining possibility to apply claimed pharmaceutical compositions based on claimed compound for prevention and treatment of inflammatory, bronchopulmonary (bronchitis, pneumonia, bronchial asthma) diseases, tuberculosis.

4 cl, 10 tbl, 11 ex

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RU 2 448 961 C1

Authors

Sernov Lev Nikolaevich

Skachilova Sofija Jakovlevna

Zheltukhin Nikolaj Konstantinovich

Proskurina Oksana Vladimirovna

Mitrokhin Nikolaj Mikhajlovich

Shilova Elena Vladimirovna

Sukhanova Svetlana Alekseevna

Sernova Aleksandra L'Vovna

Shramov Dmitrij Vital'Evich

Dates

2012-04-27Published

2011-02-03Filed