BENZIMIDAZOLYLPYRIDYL ESTER SALTS AND COMPOSITIONS CONTAINING THEM Russian patent published in 2012 - IPC C07D401/14 A61K31/4439 A61P35/00 

Abstract RU 2457206 C2

FIELD: medicine, pharmaceutics.

SUBSTANCE: present invention refers to {1-methyl-5-[2-(5-trifluoromethyl-1H-imidazol-2-yl)pyridin-4-yloxy]-1H-benzimidazol-2-yl}(4-trifluoromethylphenyl)amine salt. Also, the invention refers to a pharmaceutical composition based on the declared salt, to a method for preparing said pharmaceutical composition and to a method of treating cancer and/or angiogenesis based on the use of the declared salt.

EFFECT: there are prepared new {1-methyl-5-[2-(5-trifluoromethyl-1H-imidazol-2-yl)pyridine-4-yloxy]-1H-benzimidazol-2-yl}(4-trifluoromethylphenyl)amine salts showing effective biological properties.

42 cl, 12 dwg, 10 tbl, 7 ex

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RU 2 457 206 C2

Authors

Gullapalli Rampurna

Khashash Akhmad

Karpinski P'Otr Kh.

Lin' Kanvehn' L.

Lezer Ehrik M.

Okkhamafe Ogastus O.

Satton Pol Allen

Saj Ehduardo

Dates

2012-07-27Published

2007-08-30Filed