AMINE DERIVATIVE POSSESSING NPY-Y5 RECEPTOR ANTAGONIST ACTIVITY, AND APPLICATION THEREOF Russian patent published in 2012 - IPC A61K31/18 A61K31/136 A61K31/4184 A61K31/425 A61K31/428 A61P3/04 

Abstract RU 2460523 C2

FIELD: medicine.

SUBSTANCE: present invention refers to pharmaceutics, medicine and organic chemistry and concerns compounds of formulae presented below, as well as a pharmaceutical composition exhibiting NPY Y5 receptor antagonist activity, or an anorectic composition or an anti-obesity composition containing the compound of formulae presented below

EFFECT: what is presented is an amine derivative possessing npy y5 antagonist activity, and application thereof.

5 cl, 1 dwg, 2 tbl, 3 ex

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RU 2 460 523 C2

Authors

Okuno Takajuki

Koujama Naoki

Sakagami Masakhiro

Dates

2012-09-10Published

2008-10-23Filed