β-LACTAMYL-SUBSTITUTED ANALOGUES OF PHENYLALANINE, CYSTEINE AND SERINE AS VASOPRESSIN ANTAGONISTS Russian patent published in 2012 - IPC C07D205/08 C07D413/04 C07D413/14 A61K31/422 A61K31/397 A61P25/00 A61P25/24 

FIELD: chemistry.

SUBSTANCE: invention relates to compound of formula , where A, Q, R¹, R², R³, R⁴, R⁵' are represented in i.1 of the formula, as well as to its hydrates, solvates and pharmaceutically acceptable salts, Also described are application of said compound and pharmaceutical composition, including such compound, for treatment of disease condition in mammals, which is sensitive to action of antagonists of vasopressin V_1a, V_1b or V₂ receptors.

EFFECT: increase efficiency of compound application.

20 cl, 13 ex, 1 dwg