V1A-RECEPTORS AGONISTS Russian patent published in 2017 - IPC C07K7/06 C07K7/16 A61K38/11 A61P1/16 A61P9/02 

Abstract RU 2634617 C2

FIELD: pharmacology.

SUBSTANCE: invention relates to compounds of formula (I)

,

their salts, pharmaceutical compositions, and their use as vasopressin V1a-receptor agonists in the treatment of, for example, complications of cirrhosis, including bacterial peritonitis, HRS2 (type II hepatorenal syndrome) and refractory ascites.

EFFECT: increased efficiency of composition application.

39 cl, 3 tbl

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RU 2 634 617 C2

Authors

Visnevski Kazimezh

Kharris Dzheffri S.

Galyan Robert Feliks

Dates

2017-11-02Published

2013-05-09Filed