PHARMACEUTICAL COMPOSITION FOR PREVENTING AND TREATING PAROXYSMAL CONDITIONS Russian patent published in 2012 - IPC A61K31/4412 A61K47/48 A61P25/08 

Abstract RU 2469722 C1

FIELD: medicine.

SUBSTANCE: pharmaceutical composition contains a biologically active substance presented by 2-ethyl-6-methyl-3-oxypyridine succinate sorbed on a polymer carrier which is presented by polybutylcyanoacrylate nanoparticles or lactic and glycolic acid copolymer nanoparticles, and pharmaceutically acceptable substances in the following proportions, wt %: polymer carrier - 0.1-10, 2-ethyl-6-methyl-3-oxypyridine succinate - 0.1-5, excipients - the rest.

EFFECT: composition is high-effective in treating paroxysmal conditions; it has mild side effects.

6 tbl, 8 ex

Similar patents RU2469722C1

Title Year Author Number
4-BENZOYLPYRIDINE OXIME DERIVATIVES HAVING ANTICONVULSANT ACTIVITY AS AGENTS FOR TREATMENT OF EPILEPSY AND PAROXYSMAL STATES 2016
  • Durnev Andrej Dmitrievich
  • Voronina Tatyana Aleksandrovna
  • Litvinova Svetlana Aleksandrovna
  • Nerobkova Lyubov Nikolaevna
  • Gajdukov Igor Olegovich
  • Gudasheva Tatyana Aleksandrovna
  • Zhmurenko Lyudmila Aleksandrovna
  • Mokrov Grigorij Vladimirovich
RU2643091C2
DIBENZOFURAN OXIME DERIVANTS WITH ANTICONVULSANT AND NEUROPROTECTIVE ACTIVITY 2018
  • Voronina Tatyana Aleksandrovna
  • Litvinova Svetlana Aleksandrovna
  • Kutepova Inga Sergeevna
  • Nerobkova Lyubov Nikolaevna
  • Zhmurenko Lyudmila Aleksandrovna
  • Mokrov Grigorij Vladimirovich
  • Gudasheva Tatyana Aleksandrovna
  • Durnev Andrej Dmitrievich
RU2744758C2
COUMARIN, THIOCOUMARIN AND QUINOLINONE DERIVATIVES, HAVING ANTICONVULSANT ACTIVITY 2017
  • Mokrov Grigorij Vladimirovich
  • Litvinova Svetlana Aleksandrovna
  • Nerobkova Lyubov Nikolaevna
  • Kovalev Ivan Georgievich
  • Gudasheva Tatyana Aleksandrovna
  • Voronina Tatyana Aleksandrovna
  • Durnev Andrej Dmitrievich
  • Seredenin Sergej Borisovich
RU2720510C2
PHARMACEUTICAL COMPOSITION CONTAINING PHYSIOLOGICALLY ACTIVE HEPTAPEPTIDES, HAVING ANTISPASMODIC, ANXIOLYTIC, CENTRAL ANTI-INFLAMMATORY AND ANALGESIC ACTIVITY, AS WELL AS ANTI-ALCOHOL ACTIVITY 2012
  • Emel'Janova Tat'Jana Georgievna
  • Guzevatykh Ljudmila Sergeevna
  • Voronina Tat'Jana Aleksandrovna
  • Gel'Perina Svetlana Ehmmanuilovna
  • Balaban'Jan Vadim Jur'Evich
  • Ul'Janov Andrej Mikhajlovich
RU2506269C1
DERIVATIVES OF 4-PHENYLPYRROLIDONE WITH ANTICONVULSANT AND NOOTROPIC ACTIVITY AS MEANS OF TREATING EPILEPSY AND PAROXYSMAL CONDITIONS 2017
  • Voronina Tatyana Aleksandrovna
  • Kovalev Ivan Georgievich
  • Litvinova Svetlana Aleksandrovna
  • Nerobkova Lyubov Nikolaevna
  • Zhmurenko Lyudmila Aleksandrovna
  • Mokrov Grigorij Vladimirovich
  • Gudasheva Tatyana Aleksandrovna
  • Durnev Andrej Dmitrievich
RU2748419C2
SUBLINGUAL FORM OF 6-METHYL-2-ETHYL-3-HYDROXYPYRIDINE AND USING IT AS AGENT POSSESSING STIMULATING, ANORECTIC, ANTIDEPRESSANT, ANXIOLYTIC, ANTIHYPOXIC, ANTIAMNESTIC (NOOTROPIC), AND ANTIALCOHOL ACTIVITY 2012
  • Balaban'Jan Vadim Jur'Evich
  • Voronina Tat'Jana Aleksandrovna
  • Julina Elena Vladimirovna
  • Fomina Evgenija Geronievna
RU2527342C2
METHOD OF DETECTING ANTICONVULSANT ACTION OF SODIUM CITICOLINE AND VALPROATE WHEN APPLYING THEM TOGETHER ON MODEL OF ACUTE GENERALIZED CONVULSIONS CAUSED BY PENTYLENETETRAZOLE IN WISTAR MALE RATS 2015
  • Zinkovskij Konstantin Aleksandrovich
  • Zinkovskij Aleksandr Konstantinovich
  • Karpova Margarita Nikolaevna
  • Morozov Sergej Georgievich
  • Kuznetsova Lada Vladimirovna
  • Klishina Natalya Yurevna
RU2600477C1
PARENTERAL COMPOSITION CONTAINING CARBAMAZEPINE IN FORM OF SUBMICRON EMULSION POSSESSING ANTICONVULSANT ACTIVITY 2012
  • Suslina Zinaida Aleksandrovna
  • Sejfulla Roshen Dzhafarovich
  • Prokhorov Denis Igorevich
  • Voronina Tat'Jana Aleksandrovna
  • Kaplun Aleksandr Petrovich
  • Kapitsa Inga Gennad'Evna
  • Zhuravko Anastasija Sergeevna
  • Abaimov Denis Aleksandrovich
  • Sariev Abrek Kuangalievich
RU2490016C1
4-(3,4-DIBROMOTHIOPHENE CARBONYL)-2,6,8,12-TETRAACETYL-2,4,6,8,10,12-HEXAAZATETRACYCLO[5,5,0,0,0]DODECANE USED AS AN ANTICONVULSANT 2018
  • Krylova Svetlana Gennadevna
  • Poveteva Tatyana Nikolaevna
  • Sysolyatin Sergej Viktorovich
  • Suslov Nikolaj Innokentevich
  • Zueva Elena Petrovna
  • Nesterova Yuliya Vladimirovna
  • Afanaseva Olga Gennadevna
  • Lopatina Kseniya Aleksandrovna
  • Kulpin Pavel Valerevich
  • Zhdanov Vadim Vadimovich
  • Kulagina Darya Aleksandrovna
  • Malykhin Valerij Viktorovich
  • Vorozhtsov Aleksandr Borisovich
RU2684107C1
ANTICONVULSANT AND METHOD FOR PREPARING IT 2013
  • Leonidov Nikolaj Borisovich
  • Jakovlev Ruslan Jur'Evich
  • Lisichkin Georgij Vasil'Evich
RU2508098C1

RU 2 469 722 C1

Authors

Avakjan Gagik Norajrovich

Avakjan Georgij Gagikovich

Balaban'Jan Vadim Jur'Evich

Voronina Tat'Jana Aleksandrovna

Nerobkova Ljubov' Nikolaevna

Dates

2012-12-20Published

2011-05-20Filed