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(19)

RU

(11)

2 470 021

(13)

C2

(51)

IPC

C07D401/12(2006-01-01)

C07D401/14(2006-01-01)

C07D413/14(2006-01-01)

C07D417/14(2006-01-01)

A61K31/4525(2006-01-01)

A61K31/454(2006-01-01)

A61K31/4535(2006-01-01)

A61P25/00(2006-01-01)

(21) (22)

Application

2009147733/04, 2008-05-22

(24)

Start date

2008-05-22

(22)

Actual filing date

2008-05-22

(45)

Published

2012-12-20

(72)

Inventor

Breslin Majkl Dzh.Koulman Pol Dzh.Koks Kristofer D.Shrajer Dzhon D.

(73)

Holder

Merk Sharp Ehnd Domeh Korp.

PYRIDYL-PIPERIDINE ANTAGONISTS OF OREXIN RECEPTORS Russian patent published in 2012 - IPC C07D401/12 C07D401/14 C07D413/14 C07D417/14 A61K31/4525 A61K31/454 A61K31/4535 A61P25/00 

Abstract RU 2470021 C2

FIELD: medicine, pharmaceutics.

SUBSTANCE: claimed invention describes specific compounds, namely pyridyl-piperidine compounds, which represent antagonists of orexin receptors and can be used for treatment or prevention of neurologic and psychiatric disorders and diseases, in development of which orexin receptors participate.

EFFECT: claimed invention relates to pharmaceutical compositions, containing said compounds, as well as to application of said compounds and compositions for prevention or treatment of diseases, in development of which orexin receptors participate.

5 cl, 1 ex, 2 tbl

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RU 2 470 021 C2

Authors

Breslin Majkl Dzh.

Koulman Pol Dzh.

Koks Kristofer D.

Shrajer Dzhon D.

Dates

2012-12-20—Published

2008-05-22—Filed

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