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(19)

(11)

2 458 924

(13)

(51)

IPC

C07D401/14(2006-01-01)

C07D403/14(2006-01-01)

C07D413/14(2006-01-01)

C07D471/04(2006-01-01)

C07D487/04(2006-01-01)

C07D491/48(2006-01-01)

C07D491/52(2006-01-01)

C07D495/04(2006-01-01)

A61K31/551(2006-01-01)

A61P3/04(2006-01-01)

A61P25/20(2006-01-01)

(21) (22)

Application

2009125024/04, 2007-11-30

(24)

Start date

2007-11-30

(22)

Actual filing date

2007-11-30

(45)

Published

2012-08-20

(72)

Inventor

Bergman Dzheffri M.Breslin Majkl Dzh.Koulman Pol Dzh.Koks Kristofer D.Merser Svati P.Roker Ehntoni Dzh.

(73)

Holder

Merk Sharp Ehnd Domeh Korp.

DIAZEPANE SUBSTITUTED COMPOUNDS AS OREXIN RECEPTOR ANTAGONISTS Russian patent published in 2012 - IPC C07D401/14 C07D403/14 C07D413/14 C07D471/04 C07D487/04 C07D491/48 C07D491/52 C07D495/04 A61K31/551 A61P3/04 A61P25/20

Abstract RU 2458924 C2

FIELD: medicine, pharmaceutics.

SUBSTANCE: there are produced new diazepane substituted compounds representing various heterocyclic systems, including condensed, pharmaceutical compositions containing said compounds.

EFFECT: producing the compounds and compositions for preventing and treating neurological and mental disorders and diseases with involved orexin receptors.

13 cl, 1 tbl

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RU 2 458 924 C2

Authors

Bergman Dzheffri M.

Breslin Majkl Dzh.

Koulman Pol Dzh.

Koks Kristofer D.

Merser Svati P.

Roker Ehntoni Dzh.

Dates

2012-08-20—Published

2007-11-30—Filed