CRYSTALS OF PRASUGREL HYDROBROMATE Russian patent published in 2013 - IPC C07D495/04 A61K31/4365 A61P7/02 

Abstract RU 2484094 C1

FIELD: medicine.

SUBSTANCE: invention describes crystals of 2-acetoxy-5-(α-cyclopropylcarbonyl-2-fluorobenzyl)-4,5,6,7-tetrahydrothieno[3,2-c]pyridine (prasugrel) hydrobromate, comprisions of crystals and pharmaceutical compositions containing them for preventing and treating the diseases associated with thrombus or embolism in an animal.

EFFECT: there are prepared new crystals of prasugrel hydrobromate which possess improved stability and solubility, and can find application in medicine.

13 cl, 7 dwg, 3 tbl, 11 ex

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RU 2 484 094 C1

Authors

Juan' Chzhehdun

Chehn Sindong

Jan Julej

Tun Lin

Juj Sjun

Chzhan Lajfan

Chzhou Vehnlian

Dates

2013-06-10Published

2010-03-31Filed