BENZYL DERIVATIVES OF GLYCOSIDES AND METHODS OF THEIR APPLICATION Russian patent published in 2013 - IPC C07G3/00 A61K31/70 C07H7/04 A61P3/00 A61K31/35 

Abstract RU 2492175 C2

FIELD: medicine, pharmaceutics.

SUBSTANCE: invention also relates to pharmaceutical compositions. Compounds of the formula given below are used for treatment of diabetes mellitus of type 1 or type 2, hyperglycemia, diabetic complications, insulin-resistance, metabolic syndrome, hyperinsulinemia, hypertension, obesity, edema, dislipidemia, chronic heart failure, atherosclerosis or related diseases, and can be introduced simultaneously or successively with at least one additional therapeutic agent, selected from group consisting of anti-diabetes agent, agent, which reduces content of lipids/modulates lipids, agent for treatment of diabetic complications, anti-obesity agent, hypotensive agent, anti-hyperuricemia agent and agent for treatment of chronic heart failure, atherosclerosis or related diseases.

EFFECT: claimed are compounds which possess inhibiting action on sodium-dependent co-carrier of glucose SGLT.

8 cl, 50 ex, 1 tbl, 15 dwg

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RU 2 492 175 C2

Authors

Chehn' Juan'Vehj

Fehn Jan'

Sjuj Bajkhua

Lv Binkhua

Sid Brajan

Khehd Majkl Dzh.

Chehn Khuavehj

Chehn Tszelin

Sjuj Min

Van Tsunna

Du Tszian'

Chzhan Lili

Sjuj Geh

U Juehlin'

Dates

2013-09-10Published

2008-04-01Filed