THIENOPYRIDAZINE COMPOUNDS, PREPARING THEM, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM, AND USING THEM Russian patent published in 2013 - IPC C07D495/04 A61K31/5025 A61K31/381 A61P35/00 

Abstract RU 2494103 C2

FIELD: medicine, pharmaceutics.

SUBSTANCE: invention refers to thienopyridazine compounds of formula (I) and to pharmaceutically acceptable salts and hydrates thereof, wherein R1 and R2 independently mean H or C1-4 alkyl; R3 means a saturated or unsaturated 5- or 6-members ring containing N, S or O, or optical isomers thereof, R4 means phenyl, monosubstituted or disubstituted halogen. The invention also refers to a method for preparing the above compounds and to a pharmaceutical composition for treating and preventing tumour diseases containing the above compounds.

EFFECT: there are prepared new compounds that may be used in medicine for treating anti-tumour diseases, particularly cancer.

12 cl, 3 tbl, 19 ex

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RU 2 494 103 C2

Authors

Vu Chzhanguj

Dates

2013-09-27Published

2009-01-07Filed