AMINO ACID DERIVATIVES Russian patent published in 2013 - IPC C07C233/49 C07C235/34 C07C255/57 C07C279/14 C07C323/59 C07D207/452 C07D209/20 C07D307/85 C07D311/12 C07D405/06 A61K31/198 A61K31/216 A61K31/27 A61K31/277 A61K31/343 A61K31/37 A61K31/4015 A61K31/405 A61P29/02 

Abstract RU 2499790 C2

FIELD: chemistry.

SUBSTANCE: amino acid derivatives form new compounds of a common formula (I) with radicals values indicated in description. Amino acid derivatives disclosed herein are novel compounds which demonstrate excellent analgesic activity not only with respect to nociceptive pain model animals, but also with respect to neuropathic pain model animals.

EFFECT: amino acid derivatives medical are very effective as medicinal agents for treatment of various diseases accompanied by pain.

19 cl, 175 ex, 15 tbl

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RU 2 499 790 C2

Authors

Ookubo Tomokhiro

Nakamura Ko

Nanba Khirojosi

Josida Khirojuki

Nakadzava Jositaka

Dates

2013-11-27Published

2009-09-17Filed