NOVEL ANTIBACTERIAL MEDICATIONS FOR TREATMENT OF GRAM-POSITIVE INFECTIONS Russian patent published in 2014 - IPC C07D403/12 C07K7/50 A61K31/4045 A61K38/08 A61P31/04 

Abstract RU 2512396 C2

FIELD: chemistry.

SUBSTANCE: invention relates to novel lipopeptide compound of formula (I) , and to its pharmaceutically acceptable salts, where: R represents: and v represents integer number from 3 to 5. Invention also relates to based on the claimed compound pharmaceutical composition, which possesses antibacterial activity.

EFFECT: obtained is novel compound of formula (I), which can be applied in medicine in form of antibacterial medications against Clostridium difficile.

26 cl, 9 tbl, 20 ex

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RU 2 512 396 C2

Authors

Pirson Andre Li

Metkaf Chester A Iii

Li Tszin

Dates

2014-04-10Published

2009-12-18Filed