METHOD OF OBTAINING 4-AMINO-5-FLUORO-3-HALOGEN-6-(SUBSTITUTED)PICOLINATES Russian patent published in 2015 - IPC C07D213/04 A01N43/40 A01P13/02 

Abstract RU 2545074 C1

FIELD: chemistry.

SUBSTANCE: invention relates to method of obtaining 4-amino-5-fluoro-3-halogen-6-(substituted)picolinate of formula I , where W represents Cl, Br or I; R represents C1-C4 alkyl, cyclopropyl, C2-C4 alkenyl or phenyl, substituted with 1-4 substituents, independently selected from halogen, C1-C4 alkyl, C1-C4 halogenalkyl, C1-C4 alkoxy or C1-C4 halogenalkoxy; and R1 represents C1-C12 alkyl or non-substituted C7-C11 arylalkyl; which includes the following stages: fluorine exchange, amination, halogen exchange, halogenation and binding by means of transition metal.

EFFECT: method improvement.

7 cl, 6 ex

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RU 2 545 074 C1

Authors

Uajteker Gregori T.

Arndt Kim Eh.

Renga Dzhejms M.

Chzhu Juan'Min

Lou Kristian T.

Siddall Tomas L.

Podkhores Dehvid E.

Rot Gari Alan

Vest Skott P.

Dates

2015-03-27Published

2012-01-24Filed