NEW OCTAPEPTIDE COMPOUNDS REPRESENTING SOMATOSTATIN DERIVATIVES Russian patent published in 2015 - IPC C07K7/64 C07K14/655 A61K38/08 A61K38/31 A61P5/02 

Abstract RU 2547940 C2

FIELD: medicine, pharmaceutics.

SUBSTANCE: invention refers to biotechnology and medicine. A compound (I) has an affinity to some subtypes of somatostatin receptors, and therefore can be used as a therapeutically active peptide in developing formulations of therapeutic agents for treating pathological conditions or diseases, which involve one or more somatostatin receptors. Besides, the compound (I) can be used as a peptide used as a carrier in prescription formulations.

EFFECT: what is presented is a new octapeptide compound of general formula (I): H-2-Nal1-cyclo(Cys2-Tyr3-AA4-Lys5-Val6-Cys7)-Thr8-NH2.

20 cl, 3 tbl, 25 ex

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Authors

Paternostr Mari-Terez

Sentra Zhan-Kristof

Valeri Selin

Ru Stefan

Russo Bernar

Ehjsselstejn Marten

Sherif-Shejkkh Rolan

Artzner Frank

Dates

2015-04-10Published

2009-09-29Filed