FIELD: medicine, pharmaceutics.
SUBSTANCE: invention refers to biotechnology and medicine. A compound (I) has an affinity to some subtypes of somatostatin receptors, and therefore can be used as a therapeutically active peptide in developing formulations of therapeutic agents for treating pathological conditions or diseases, which involve one or more somatostatin receptors. Besides, the compound (I) can be used as a peptide used as a carrier in prescription formulations.
EFFECT: what is presented is a new octapeptide compound of general formula (I): H-2-Nal1-cyclo(Cys2-Tyr3-AA4-Lys5-Val6-Cys7)-Thr8-NH2.
20 cl, 3 tbl, 25 ex
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Authors
Dates
2015-04-10—Published
2009-09-29—Filed