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(19)

RU

(11)

2 595 525

(13)

C2

(51)

IPC

C07K7/06(2006-01-01)

C07K14/655(2006-01-01)

A61K38/08(2006-01-01)

A61P5/02(2006-01-01)

(21) (22)

Application

2013102588/04, 2011-06-21

(24)

Start date

2011-06-21

(22)

Actual filing date

2011-06-21

(45)

Published

2016-08-27

(72)

Inventor

Sentra Zhan-KristofLigeti MelindaRusso BernarArtzner FrankTarabu KristofPaternostr Mari-TerezFej NikolyaSherif-Shejkkh RolanValeri Selin

(73)

Holder

Ipsen Farma S.A.S.Kommissariat A L'Enerzhi AtomikSantr Nasonal De Lya Reshersh Sentifik

NEW OCTAPEPTIDE COMPOUNDS AND THEIR THERAPEUTIC APPLICATION Russian patent published in 2016 - IPC C07K7/06 C07K14/655 A61K38/08 A61P5/02 

Abstract RU 2595525 C2

FIELD: pharmaceutics.

SUBSTANCE: invention relates to novel octapeptide compounds of general formula (I), which have high affinity to some subtypes of somatostatin receptors. Invention also relates to pharmaceutical compositions containing said products and use thereof for preparing a drug R-AA1-cyclo-(AA2-Tyr3-D-TRP4-AA5-Val6-Cys7)-Thr8-NH2 (I).

EFFECT: compounds are intended for treating pathological conditions or diseases, involving one or more somatostatin receptors.

17 cl, 9 ex

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RU 2 595 525 C2

Authors

Sentra Zhan-Kristof

Ligeti Melinda

Russo Bernar

Artzner Frank

Tarabu Kristof

Paternostr Mari-Terez

Fej Nikolya

Sherif-Shejkkh Rolan

Valeri Selin

Dates

2016-08-27—Published

2011-06-21—Filed

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