ARALKYL BENSYL ETHERS, METHODS OF SYNTHESIS THEREOF, INTERMEDIATE COMPOUNDS AND THEIR USE, METHODS FOR TREATMENT AND/OR PREVENTION, PHARMACEUTICAL COMPOSITION AND DRUG ON BASIS OF THESE COMPOUNDS Russian patent published in 2015 - IPC C07D233/60 C07D401/12 C07C22/04 A61K31/4174 A61K31/4178 A61P31/04 A61P31/10

Abstract RU 2548009 C2

FIELD: chemistry.

SUBSTANCE: invention relates to organic chemistry, specifically to bensyl aralkyl ether of formula or to its pharmaceutically acceptable salt, where: Ar represents imidazolil; R₁, R₂, R₄ and R₅ independently stand for hydrogen; R₃ stands for a halogen; R₆ stands for trifluoromethyl or trichloromethyl; n is an integer from 0 to 2; and m is 1. The invention also relates to the use of the compound of formula (1) for the treatment and/or prevention of diseases caused by fungi, or bacteria.

EFFECT: obtained new heterocyclic compounds with useful biological properties.

4 cl, 4 dwg, 9 tbl, 8 ex

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RU 2 548 009 C2

Authors

Keppler Artur Franz

Zaim Marcio Henrique

Dates

2015-04-10—Published

2010-08-27—Filed