DERIVATIVES OF TRICYCLIC INDOLE AS PBR LIGANDS Russian patent published in 2015 - IPC C07D209/80 C07D209/88 A61K49/06 A61K51/04 

Abstract RU 2551423 C2

FIELD: chemistry.

SUBSTANCE: invention relates to a radioindicator for PET, which possesses improved properties with respect to visualisation of peripheral benzodiazepine receptors (PBR) in comparison with known radioindicators for PET. In accordance with the claimed invention also claimed are: a predecessor compound for obtaining the radioindicator for PET in accordance with the invention and methods of obtaining the said predecessor compound and the said radioindicator for PET.

EFFECT: claimed is a radiopharmaceutical composition, containing the radioindicator for PET in accordance with the invention and methods for the application of the radioindicator for PET and the radiopharmaceutical composition .

23 cl, 8 dwg, 12 ex

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Authors

Achanath Randha

Balaji Srinath

Fairway Steven Michael

Mantzilas Dimitrios

Mokkapati Umamaheshwar

O'Shea Dennis

Passmore Joanna Marie

Shan Bo

Trigg William John

Wadsworth Harry John

Kadavilpparampu Mohamed Afsal Mohammed

Dates

2015-05-27Published

2011-03-28Filed