METHODS OF MODULATING ACTIVITY OF MC5 RECEPTOR AND TREATMENT OF CONDITIONS RELATED TO THEREOF Russian patent published in 2015 - IPC A61K31/551 C07D401/06 C07D409/12 C07D401/12 C07D413/12 A61P17/10 A61P17/08

Abstract RU 2555343 C9

FIELD: medicine, pharmaceutics.

SUBSTANCE: invention relates to field of pharmaceutics, namely, deals with compounds of formula , suitable for reduction of regulation of biological activity of melanocortin-5 receptor (MC5R). Such diseases and/or conditions include, but are not limited by, acne, seborrhoea, seborrheic dermatitis, cancer and inflammatory diseases.

EFFECT: compounds of claimed invention can be applied for treatment of diseases and/or conditions, in which reducing regulation of MC5R is favourable.

3 cl, 109 ex, 7 tbl

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RU 2 555 343 C9

Authors

Blaskovich Mark Arnol'D Tomas

Kehssidi Piter Dzhozef

Dates

2015-07-10—Published

2009-02-27—Filed