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(19)

RU

(11)

2 557 242

(13)

C2

(51)

IPC

C07D471/04(2006-01-01)

C07D487/04(2006-01-01)

C07D498/14(2006-01-01)

C07D241/00(2006-01-01)

A61K31/498(2006-01-01)

A61P35/00(2006-01-01)

(21) (22)

Application

2012121806/04, 2010-10-22

(24)

Start date

2010-10-22

(22)

Actual filing date

2010-10-22

(45)

Published

2015-07-20

(72)

Inventor

Kharris Roj L.Sapienza DzhonShevlin GraziehllaPapa PatrikLi Brenden DzhingsiPakard GarrikChzhao TszintszinDzhokil Patrik EhntoniMortensen DeboraRiggs DzhenniferGamboa Khuan AntonioBosham Mehri DzhordzhKrejlejn Mehtt'Ju MajklKotare Mokhit AtulPerren-Ninkovich SofiPaj FilipLeong Uill'Jam Vehj-KhvaEhl'Sner JanChoudkhuri Anusuja

(73)

Holder

Signal Farmas'Jutikalz, Ehlehlsi

METHODS OF OBTAINING AND PURIFICATION OF HETEROARYL COMPOUNDS Russian patent published in 2015 - IPC C07D471/04 C07D487/04 C07D498/14 C07D241/00 A61K31/498 A61P35/00 

Abstract RU 2557242 C2

FIELD: medicine, pharmaceutics.

SUBSTANCE: invention relates to methods of obtaining heteroaryl compounds, represented by structural formulae (I) or (II): where R1-R4 have values, given in subcl. 1,14 of the formula.

EFFECT: compounds can be used for treatment or prevention of cancer, inflammatory states, immunological states, etc.

29 cl, 20 ex

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RU 2 557 242 C2

Authors

Kharris Roj L.

Sapienza Dzhon

Shevlin Graziehlla

Papa Patrik

Li Brenden Dzhingsi

Pakard Garrik

Chzhao Tszintszin

Dzhokil Patrik Ehntoni

Mortensen Debora

Riggs Dzhennifer

Gamboa Khuan Antonio

Bosham Mehri Dzhordzh

Krejlejn Mehtt'Ju Majkl

Kotare Mokhit Atul

Perren-Ninkovich Sofi

Paj Filip

Leong Uill'Jam Vehj-Khva

Ehl'Sner Jan

Choudkhuri Anusuja

Dates

2015-07-20—Published

2010-10-22—Filed

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