ANTIRETROVIRAL AGENTS BASED ON AZIDOTHYMIDINE DERIVATIVES Russian patent published in 2015 - IPC C07D321/00 A61K31/506 A61P31/18 

Abstract RU 2561501 C1

FIELD: chemistry.

SUBSTANCE: invention relates to antiretroviral azidothymidine derivatives of formula 1 and can be used as a medicinal agent. , where: R1+R2=-CH2(CH2)2CH2-, R1+R2=-CH2(CH2)3CH2-, R1=H, R2=CH3, R1=H, R2=CH2CH2CH3, R1=H, R2=C(CH3)3, R1=H, R2=CH2(CH2)6CH3.

EFFECT: novel effective agents with low toxicity against retroviral infections.

16 ex, 2 tbl

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Authors

Shtyrlin Jurij Grigor'Evich

Pavel'Ev Roman Sergeevich

Khajrullina Regina Rishatovna

Rizvanov Al'Bert Anatol'Evich

Martynova Ekaterina Vladimirovna

Dates

2015-08-27Published

2014-08-05Filed